94
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MedChemExpress
gne 781 Gne 781, supplied by MedChemExpress, used in various techniques. Bioz Stars score: 94/100, based on 1 PubMed citations. ZERO BIAS - scores, article reviews, protocol conditions and more https://www.bioz.com/product/gne-781/GNE-781/pmc11167439-30-0-2 Average 94 stars, based on 1 article reviews
gne 781 - by Bioz Stars,
2026-09
94/100 stars
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GNE-781(CAT: I011859) is an orally active, highly potent, and selective bromodomain inhibitor targeting the CREB-binding protein (CBP), exhibiting an IC50 of 0.94 nM in TR-FRET assays. It shows strong cellular activity with minimal off-target effects,
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90
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Genentech inc
cbp/ep300 bromodomain inhibitors gne-781 Cbp/Ep300 Bromodomain Inhibitors Gne 781, supplied by Genentech inc, used in various techniques. Bioz Stars score: 90/100, based on 1 PubMed citations. ZERO BIAS - scores, article reviews, protocol conditions and more https://www.bioz.com/product/gne-781/gne+781/pm40156557-67-10-25 Average 90 stars, based on 1 article reviews
cbp/ep300 bromodomain inhibitors gne-781 - by Bioz Stars,
2026-09
90/100 stars
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N/A
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A selective inhibitor of the bromodomain of Cyclic adenosine monophosphate Response Element Binding protein Binding Protein (CREBBP or CBP) with anti-tumoral activity. The CBP inhibition regulates oncogene MYC and impairs differentiation of regulatory T cells..
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InformationGNE-781 GNE-781 (compound 19) is an orally active, highly potent and selective bromodomain inhibitor of cyclic adenosine monophosphate response element binding protein (CBP) with IC50 of 0.94 nM in TR-FRET assay. GNE-781 also inhibits BRET
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