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MedChemExpress diltiazem
Loading doses, infusion rates, formulations, and microdialysis probe recoveries used for the 14 compounds in rat microdialysis study ( n = 3, mean ± SD)
Diltiazem, supplied by MedChemExpress, used in various techniques. Bioz Stars score: 94/100, based on 1 PubMed citations. ZERO BIAS - scores, article reviews, protocol conditions and more
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Loading doses, infusion rates, formulations, and microdialysis probe recoveries used for the 14 compounds in rat microdialysis study ( n = 3, mean ± SD)

Journal: Pharmacology Research & Perspectives

Article Title: Effects of membrane transport activity and cell metabolism on the unbound drug concentrations in the skeletal muscle and liver of drugs: A microdialysis study in rats

doi: 10.1002/prp2.879

Figure Lengend Snippet: Loading doses, infusion rates, formulations, and microdialysis probe recoveries used for the 14 compounds in rat microdialysis study ( n = 3, mean ± SD)

Article Snippet: Antipyrine, ofloxacin, lamotrigine, digoxin, quinidine, atenolol, carbamazepine, propranolol, diltiazem, memantine, diphenhydramine, pyrilamine, and gabapentin were purchased from MedChemExpress (Monmouth Junction).

Techniques: Formulation

Pharmacokinetic parameters of the 14 compounds following an IV single bolus ( n = 3; mean ± SD) ( n = 3, mean ± SD)

Journal: Pharmacology Research & Perspectives

Article Title: Effects of membrane transport activity and cell metabolism on the unbound drug concentrations in the skeletal muscle and liver of drugs: A microdialysis study in rats

doi: 10.1002/prp2.879

Figure Lengend Snippet: Pharmacokinetic parameters of the 14 compounds following an IV single bolus ( n = 3; mean ± SD) ( n = 3, mean ± SD)

Article Snippet: Antipyrine, ofloxacin, lamotrigine, digoxin, quinidine, atenolol, carbamazepine, propranolol, diltiazem, memantine, diphenhydramine, pyrilamine, and gabapentin were purchased from MedChemExpress (Monmouth Junction).

Techniques:

Steady‐state unbound drug concentrations in liver, muscle, and blood of Class I compounds with good membrane permeability that are not efflux and uptake transporter substrates ( n = 3, mean ± SD)

Journal: Pharmacology Research & Perspectives

Article Title: Effects of membrane transport activity and cell metabolism on the unbound drug concentrations in the skeletal muscle and liver of drugs: A microdialysis study in rats

doi: 10.1002/prp2.879

Figure Lengend Snippet: Steady‐state unbound drug concentrations in liver, muscle, and blood of Class I compounds with good membrane permeability that are not efflux and uptake transporter substrates ( n = 3, mean ± SD)

Article Snippet: Antipyrine, ofloxacin, lamotrigine, digoxin, quinidine, atenolol, carbamazepine, propranolol, diltiazem, memantine, diphenhydramine, pyrilamine, and gabapentin were purchased from MedChemExpress (Monmouth Junction).

Techniques: Membrane, Permeability